Publicaciones (22) Publicaciones de Carme Masdeu Margalef

2023

  1. Efficient AntiMycolata Agents by Increasing the Lipophilicity of Known Antibiotics through Multicomponent Reactions

    Antibiotics, Vol. 12, Núm. 1

  2. Gel-Free Tools for Quick and Simple Screening of Anti-Topoisomerase 1 Compounds

    Pharmaceuticals, Vol. 16, Núm. 5

  3. Synthesis of Fused Nitrogenated Heterocycles: Intramolecular Povarov Reaction

    Advances in Organic Synthesis (Bentham Science Publishers), pp. 40-111

  4. The Intramolecular Povarov Tool in the Construction of Fused Nitrogen-Containing Heterocycles

    Topics in Current Chemistry, Vol. 381, Núm. 4

2021

  1. A patent review of topoisomerase I inhibitors (2016–present)

    Expert Opinion on Therapeutic Patents, Vol. 31, Núm. 6, pp. 473-508

2020

  1. Fused 1,5-Naphthyridines: Synthetic Tools and Applications

    Molecules (Basel, Switzerland), Vol. 25, Núm. 15

  2. Synthetic strategies, reactivity and applications of 1,5-naphthyridines

    Molecules, Vol. 25, Núm. 14

2018

  1. In vitro and in vivo activity of a new small-molecule inhibitor of HDAC6 in mantle cell lymphoma

    Haematologica

  2. Recent advances of the Povarov reaction in medicinal chemistry

    Drug Discovery Today: Technologies, Vol. 29, pp. 71-79

2015

  1. Development and validation of a LC-MS assay for the quantification of ikh12 a novel anti-tumor candidate in rat plasma and tissues and its application in a pharmacokinetic study

    Biomedical Chromatography, Vol. 29, Núm. 8, pp. 1249-1258

2010

  1. Formation of γ-oxoacids and 1 H-pyrrol-2(5 H)-ones from α,β-unsaturated ketones and ethyl nitroacetate

    Journal of Organic Chemistry, Vol. 75, Núm. 21, pp. 7435-7438

2009

  1. Highly enantioselective conjugate additions of aldehydes to vinyl sulfones

    Chemistry - A European Journal, Vol. 15, Núm. 7, pp. 1562-1565

  2. Multicomponent access to functionalized mesoionic structures based on TFAA activation of isocyanides: Novel domino reactions

    European Journal of Organic Chemistry, pp. 617-625

2008

  1. Benzimidazolium salts as small, nonpeptidic and BBB-permeable human prolyl oligopeptidase inhibitors

    ChemMedChem, Vol. 3, Núm. 10, pp. 1558-1565

2007

  1. Double insertion of isocyanides into dihydropyridines: Direct access to substituted benzimidazolium salts

    Angewandte Chemie - International Edition, Vol. 46, Núm. 17, pp. 3043-3046

2006

  1. Hydro-, halo- and seleno-carbamoylation of cyclic enol ethers and dihydropyridines: New mechanistic pathways for Passerini-and Ugi-type multicomponent reactions

    QSAR and Combinatorial Science, Vol. 25, Núm. 5-6, pp. 465-473

  2. Isocyanide addition to pyridinium salts. Efficient entry into substituted nicotinonitrile derivatives

    Organic Letters, Vol. 8, Núm. 25, pp. 5789-5792

2004

  1. Straightforward α-carbamoylation of NADH-like dihydropyridines and enol ethers

    Tetrahedron Letters, Vol. 45, Núm. 42, pp. 7907-7909

2000

  1. Introduction of heteroatom-based substituents into 1,4-dihydropyridines by means of a halogen-mediated, oxidative protocol: Diamination, sulfonylation, sulfinylation, bis-sulfanylation, and halo-phosphonylation processes

    Chemistry - A European Journal, Vol. 6, Núm. 10, pp. 1763-1772

1998

  1. 'Nonbiomimetic' oxidations of dihydropyridines

    Journal of Organic Chemistry, Vol. 63, Núm. 26, pp. 10001-10005