Publicaciones en colaboración con investigadores/as de Aarhus University (12)

2023

  1. Gel-Free Tools for Quick and Simple Screening of Anti-Topoisomerase 1 Compounds

    Pharmaceuticals, Vol. 16, Núm. 5

2022

  1. Synthesis of hybrid phosphorated indenoquinolines and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry Letters, Vol. 57

2021

  1. A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors

    Sensors, Vol. 21, Núm. 14

  2. Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry, Vol. 40

  3. Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)

    Pharmaceuticals, Vol. 14, Núm. 8

  4. Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1

    Pharmaceutics, Vol. 13, Núm. 8

2020

  1. Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents

    Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861

  2. Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives

    European Journal of Medicinal Chemistry, Vol. 195

2019

  1. Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones

    European Journal of Medicinal Chemistry, Vol. 178, pp. 752-766

2018

  1. Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity

    European Journal of Medicinal Chemistry, Vol. 149, pp. 225-237

2017

  1. Advantages of an optical nanosensor system for the mechanistic analysis of a novel topoisomerase i targeting drug: A case study

    Nanoscale, Vol. 9, Núm. 5, pp. 1886-1895

2016

  1. Synthesis and biological evaluation of indeno[1,5]naphthyridines as topoisomerase i (TopI) inhibitors with antiproliferative activity

    European Journal of Medicinal Chemistry, Vol. 115, pp. 179-190