Francisco J. Palacios Gambra-rekin lankidetzan egindako argitalpenak (64)

2024

  1. Antileishmanial Effect of 1,5- and 1,8-Substituted Fused Naphthyridines

    Molecules, Vol. 29, Núm. 1

  2. Aza-Povarov Reaction. A Method for the Synthesis of Fused Tetracyclic Chromeno[4,3-d]pyrido[1,2-a]pyrimidines

    Journal of Organic Chemistry, Vol. 89, Núm. 2, pp. 1099-1107

2023

  1. Efficient AntiMycolata Agents by Increasing the Lipophilicity of Known Antibiotics through Multicomponent Reactions

    Antibiotics, Vol. 12, Núm. 1

2022

  1. Multicomponent Synthesis of Unsaturated γ-Lactam Derivatives. Applications as Antiproliferative Agents through the Bioisosterism Approach: Carbonyl vs. Phosphoryl Group

    Pharmaceuticals, Vol. 15, Núm. 5

  2. The design and discovery of topoisomerase I inhibitors as anticancer therapies

    Expert Opinion on Drug Discovery, Vol. 17, Núm. 6, pp. 581-601

2021

  1. A dual-sensor-based screening system for in vitro selection of tdp1 inhibitors

    Sensors, Vol. 21, Núm. 14

  2. A patent review of topoisomerase I inhibitors (2016–present)

    Expert Opinion on Therapeutic Patents, Vol. 31, Núm. 6, pp. 473-508

  3. Design, synthesis and cytotoxic evaluation of diphenyl(quinolin-8-yl)phosphine oxides

    Tetrahedron Letters, Vol. 70

  4. Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

    Bioorganic and Medicinal Chemistry, Vol. 40

  5. Hybrid quinolinyl phosphonates as heterocyclic carboxylate isosteres: Synthesis and biological evaluation against topoisomerase 1b (top1b)

    Pharmaceuticals, Vol. 14, Núm. 8

  6. Naphthyridine derivatives induce programmed cell death in naegleria fowleri

    Pharmaceuticals, Vol. 14, Núm. 10

  7. Simple and fast dna based sensor system for screening of small-molecule compounds targeting eukaryotic topoisomerase 1

    Pharmaceutics, Vol. 13, Núm. 8

2020

  1. Fused 1,5-Naphthyridines: Synthetic Tools and Applications

    Molecules (Basel, Switzerland), Vol. 25, Núm. 15

  2. New Challenges in Drug Discovery – July 8–11, 2019, Vitoria-Gasteiz, Spain

    ChemMedChem

  3. Novel phosphine sulphide gold(i) complexes: topoisomerase I inhibitors and antiproliferative agents

    Dalton Transactions, Vol. 49, Núm. 23, pp. 7852-7861

  4. Parasitic infectious diseases

    European Journal of Medicinal Chemistry

  5. Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives

    European Journal of Medicinal Chemistry, Vol. 195

  6. Synthetic strategies, reactivity and applications of 1,5-naphthyridines

    Molecules, Vol. 25, Núm. 14

2019

  1. Antileishmanial activity of new hybrid tetrahydroquinoline and quinoline derivatives with phosphorus substituents

    European Journal of Medicinal Chemistry, Vol. 162, pp. 18-31

  2. Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones

    European Journal of Medicinal Chemistry, Vol. 178, pp. 752-766