Synthesis, biological evaluation, and automated docking of constrained analogues of the opioid peptide H-Dmt-d-Ala-Phe-Gly-NH 2 using the 4- or 5-methyl substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one scaffold

1. De Wachter, R.
2. De Graaf, C.
3. Keresztes, A.
4. Vandormael, B.
5. Ballet, S.
6. Tóth, G.
7. Rognan, D.
8. Tourwé, D.